Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium (2022)
- Authors:
- Cruz, Luiza
- Silva, Adriana Corrêa da
- Feltrin, Clarissa
- Dichiara, Maria
- Ferrins, Lori
- Moraes, Carolina Borsoi - Universidade Federal de São Paulo (UNIFESP)
- Sjo, Peter
- Andricopulo, Adriano Defini
- Mowbray, Charles
- Oliveira, Ramon Guerra de - Universidade Estadual de Campinas (UNICAMP)
- Dessoy, Marco Aurélio - Universidade Estadual de Campinas (UNICAMP)
- Santos, Deborah Araújo dos - Universidade Estadual de Campinas (UNICAMP)
- Oliveira, Luiz Fernando Nascimento de - Universidade Estadual de Campinas (UNICAMP)
- Mollo, María Cruz - Universidade Estadual de Campinas (UNICAMP)
- Lee, Eun - Universidade Estadual de Campinas (UNICAMP)
- Duarte, Simone Michelan
- Andricopulo, Renata Krogh
- Chelucci, Rafael Consolin
- Ferreira, Leonardo Luiz Gomes
- Kratz, Jadel Muller
- Dias, Luiz Carlos - Universidade Estadual de Campinas (UNICAMP)
- USP affiliated authors: ANDRICOPULO, ADRIANO DEFINI - IFSC ; DUARTE, SIMONE MICHELAN - IFSC ; ANDRICOPULO, RENATA KROGH - IFSC ; CHELUCCI, RAFAEL CONSOLIN - IFSC ; FERREIRA, LEONARDO LUIZ GOMES - IFSC
- Unidade: IFSC
- Subjects: DOENÇAS NEGLIGENCIADAS; DOENÇA DE CHAGAS
- Keywords: Phenotypic screening; Drug Discovery; Medicinal Chemistry; Indoles; CYP51 inhibition
- Language: Inglês
- Imprenta:
- Source:
- Título do periódico: Anais eletrônicos
- Conference titles: Brazilian Symposium on Medicinal Chemistry - BrazMedChem
-
ABNT
CRUZ, Luiza et al. Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium. 2022, Anais.. Campinas: Galoá, 2022. Disponível em: https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. Acesso em: 05 jun. 2024. -
APA
Cruz, L., Silva, A. C. da, Feltrin, C., Dichiara, M., Ferrins, L., Moraes, C. B., et al. (2022). Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium. In Anais eletrônicos. Campinas: Galoá. Recuperado de https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. -
NLM
Cruz L, Silva AC da, Feltrin C, Dichiara M, Ferrins L, Moraes CB, Sjo P, Andricopulo AD, Mowbray C, Oliveira RG de, Dessoy MA, Santos DA dos, Oliveira LFN de, Mollo MC, Lee E, Duarte SM, Andricopulo RK, Chelucci RC, Ferreira LLG, Kratz JM, Dias LC. Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium [Internet]. Anais eletrônicos. 2022 ;[citado 2024 jun. 05 ] Available from: https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. -
Vancouver
Cruz L, Silva AC da, Feltrin C, Dichiara M, Ferrins L, Moraes CB, Sjo P, Andricopulo AD, Mowbray C, Oliveira RG de, Dessoy MA, Santos DA dos, Oliveira LFN de, Mollo MC, Lee E, Duarte SM, Andricopulo RK, Chelucci RC, Ferreira LLG, Kratz JM, Dias LC. Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium [Internet]. Anais eletrônicos. 2022 ;[citado 2024 jun. 05 ] Available from: https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. - Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum
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