Design, synthesis and biological activity of novel substituted 3-benzoic acid derivatives as MtDHFR inhibitors (2020)
- Authors:
- USP affiliated authors: TROSSINI, GUSTAVO HENRIQUE GOULART - FCF ; DIAS, MARCIO VINÍCIUS BERTACINE - ICB ; PARISE FILHO, ROBERTO - FCF ; FERREIRA, GLAUCIO MONTEIRO - FCF
- Unidades: FCF; ICB
- DOI: 10.1016/j.bmc.2020.115600
- Subjects: MICROBIOLOGIA; METABÓLITOS; ÁCIDOS CARBOXÍLICOS; DNA; TUBERCULOSE; CINÉTICA QUÍMICA
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Source:
- Título do periódico: Bioorganic & Medicinal Chemistry
- ISSN: 1464-3391
- Volume/Número/Paginação/Ano: v. 28, n. 15, art. 115600, 10 p., 2020
- Este periódico é de assinatura
- Este artigo NÃO é de acesso aberto
- Cor do Acesso Aberto: closed
-
ABNT
KRONENBERGER, Thales et al. Design, synthesis and biological activity of novel substituted 3-benzoic acid derivatives as MtDHFR inhibitors. Bioorganic & Medicinal Chemistry, v. 28, n. 15, p. 10 , 2020Tradução . . Disponível em: https://doi.org/10.1016/j.bmc.2020.115600. Acesso em: 06 jun. 2024. -
APA
Kronenberger, T., Ferreira, G. M., Souza, A. D. F. de, Santos, S. da S., Poso, A., Ribeiro, J. A., et al. (2020). Design, synthesis and biological activity of novel substituted 3-benzoic acid derivatives as MtDHFR inhibitors. Bioorganic & Medicinal Chemistry, 28( 15), 10 . doi:10.1016/j.bmc.2020.115600 -
NLM
Kronenberger T, Ferreira GM, Souza ADF de, Santos S da S, Poso A, Ribeiro JA, Tavares MT, Pavan FR, Trossini GHG, Dias MVB, Parise Filho R. Design, synthesis and biological activity of novel substituted 3-benzoic acid derivatives as MtDHFR inhibitors [Internet]. Bioorganic & Medicinal Chemistry. 2020 ; 28( 15): 10 .[citado 2024 jun. 06 ] Available from: https://doi.org/10.1016/j.bmc.2020.115600 -
Vancouver
Kronenberger T, Ferreira GM, Souza ADF de, Santos S da S, Poso A, Ribeiro JA, Tavares MT, Pavan FR, Trossini GHG, Dias MVB, Parise Filho R. Design, synthesis and biological activity of novel substituted 3-benzoic acid derivatives as MtDHFR inhibitors [Internet]. Bioorganic & Medicinal Chemistry. 2020 ; 28( 15): 10 .[citado 2024 jun. 06 ] Available from: https://doi.org/10.1016/j.bmc.2020.115600 - Optimization of new dihydrofolate reductase inhibitors of mycobacterium tuberculosis (mtDHFR): molecular docking, synthesis, evaluation of enzyme inhibition and antimycobacterial activity
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Informações sobre o DOI: 10.1016/j.bmc.2020.115600 (Fonte: oaDOI API)
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